Article

Prospects for the use of 3-R-benzo[f][1,2,4]triazino[2,3-d][1,4]diazepine-2,7(6H,8H)-diones as agonists and antagonists of GABAA receptors

2026-08-24

Abstract excerpt

<title>Abstract</title> Purpose The benzo[ <italic>f</italic> ][1,2,4]triazino[2,3- <italic>d</italic> ][1,4]diazepine-2,7(6 <italic>H</italic> ,8 <italic>H</italic> )-dione scaffold combines features of classical 1,4-benzodiazepines and β-carboline inverse agonists, and was therefore examined at the γ-aminobutyric acid type A receptor (GABA A R) benzodiazepine (BZD) modulatory site. Me...

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Literature Corpus work: ad194af3-c73e-50b7-bff1-b7fd05aaf0fb
DOI: 10.21203/rs.3.rs-10753552/v1

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Prospects for the use of 3-R-benzo[f][1,2,4]triazino[2,3-d][1,4]diazepine-2,7(6H,8H)-diones as agonists and antagonists of GABAA receptorsDOI 10.21203/rs.3.rs-10753552/v1Read

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