Article

Prospects for the use of 3-R-benzo[f][1,2,4]triazino[2,3-d][1,4]diazepine-2,7(6H,8H)-diones as agonists and antagonists of GABAA receptors

2026-08-26

Abstract excerpt

<title>Abstract</title> <bold>Purpose</bold> The benzo[ <italic>f</italic> ][1,2,4]triazino[2,3- <italic>d</italic> ][1,4]diazepine-2,7(6 <italic>H</italic> ,8 <italic>H</italic> )-dione scaffold combines features of classical 1,4-benzodiazepines and β-carboline inverse agonists, and was therefore examined at the γ-aminobutyric acid type A receptor (GABA A R) benzodiazepine (BZD) modula...

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Literature Corpus work: dff6382e-cfec-5bf7-9700-3071f7be9d12
DOI: 10.21203/rs.3.rs-10753552/v2

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Prospects for the use of 3-R-benzo[f][1,2,4]triazino[2,3-d][1,4]diazepine-2,7(6H,8H)-diones as agonists and antagonists of GABAA receptorsDOI 10.21203/rs.3.rs-10753552/v2Read

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