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Article

Features and potentials of ATP-site directed CK2 inhibitors.

Biochimica et biophysica acta - 30 Dec 2005

Sarno Stefania, Salvi Mauro, Battistutta Roberto, Zanotti Giuseppe, Pinna Lorenzo A

Abstract excerpt

A panel of quite specific, fairly potent and cell-permeable inhibitors of protein kinase CK2 belonging to the classes of condensed polyphenolic compounds, tetrabromobenzimidazole/triazole derivatives and indoloquinazolines have been developed, with K(i) values in the submicromolar range. Nine structures have been solved to date of complexes between the catalytic alpha subunit of CK2 and a number of these...

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Identifiers

PMID: 16198160
DOI: 10.1016/j.bbapap.2005.07.043

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PubMed metadata and Literature Corpus relationships. Corpus snapshot updated 7 Sept 2026. Manifest publication-graph-cohort-2026-09-07.1.

Source receipt: pubmed, retrieved 7 Sept 2026.

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