Article

Strain-promoted stapled peptides for inhibiting protein-protein interactions

2019-01-01

Abstract excerpt

Protein-protein interactions (PPIs) are responsible for the regulation of a variety of important functions within living organisms. Compounds which can selectively modulate aberrant PPIs are novel therapeutic candidates for treating human diseases. Whilst PPIs have traditionally been considered as ~undruggable~, research in this area has led to the emergence of several effective methodologies for targeting PPIs. O...

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Literature Corpus work: d2d6b2eb-960a-564d-8075-5b2164420c23
DOI: 10.17863/cam.35884

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