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7-Methoxy-3-Substituted-2,3,4,5-Tetrahydro-1<em>H</em>-benzo[<em>d</em>]azepin-1-ols as Prospective Radioligands for PET Imaging of the GluN2B Subunit

2026-04-13

Abstract excerpt

N-Methyl-D-aspartate (NMDA) receptors are ligand- and voltage-gated ion channels that are critical for synaptic plasticity, learning, and memory. These receptors are variously composed of GluN1, GluN2A–D, and GluN3A/B subunits. They are widely expressed in the central nervous system and are implicated in several neurological, neurodegenerative, and psychiatric disorders. The GluN2B subunit has garnered particular...

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Literature Corpus work
695341c1-a37c-50c7-98ce-6e3fcf585e47
DOI
10.20944/preprints202604.0788.v1
Open publication

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7-Methoxy-3-Substituted-2,3,4,5-Tetrahydro-1<em>H</em>-benzo[<em>d</em>]azepin-1-ols as Prospective Radioligands for PET Imaging of the GluN2B SubunitDOI 10.20944/preprints202604.0788.v1
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