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Article

Characterization of ligand-induced conformational states in the beta 2 adrenergic receptor.

Journal of receptor and signal transduction research - 1 Jan 2000

Kobilka B, Gether U, Seifert R, Lin S, Ghanouni P

Abstract excerpt

Drugs acting at G protein coupled receptors can be classified in biological assays as either agonists, partial agonists, neutral antagonists, or as inverse agonists. Very little is known about the actual molecular events and structural changes that occur in the receptor following ligand binding and during transmission of a signal across the membrane. Therefore, the structural basis for the biological...

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Methodology Data sources Editorial policy Privacy About Contact Helena Bioinformatics

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Identifiers

PMID: 10071765
DOI: 10.3109/10799899909036652

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PubMed metadata and Literature Corpus relationships. Corpus snapshot updated 7 Sept 2026. Manifest publication-graph-cohort-2026-09-07.1.

Source receipt: pubmed, retrieved 7 Sept 2026.

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