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USING DYNAMIC MASS REDISTRIBUTION TO CHARACTERISE THE PHARMACOLOGY OF THE MAS RELATED GPCR FAMILY MEMBER D (MRGPRD) RECEPTOR

2023-03-11

Abstract excerpt

Human mas-related genes such as MRGPRD are members of the seven transmembrane spanning G protein coupled receptor super family implicated in the sensation and transmission of noxious stimuli such as pain and itch, hence intervening with these may prove useful in the management of unmet patient need. To date there have been few reports of the generation of inhibitors of these receptors. To provide new tools to aid...

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Literature Corpus work: 3cf6f474-1157-5e23-868b-caa7a97140c4
DOI: 10.22541/au.167851268.89573685/v1

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