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Article

Characterization of In Vitro Synthesized Equine Metabolites of the Selective Androgen Receptor Modulators S24 and S4

2012-09-01

Abstract excerpt

Several selective androgen receptor modulators (SARMs) have been synthesized and investigated in humans, rats, and dogs in the past, but no data are yet available concerning the metabolism of SARMs in horses. The aryl-propionamide-derived drug candidates S24 and S4 (andarine) have a strong androgen receptor binding affinity and show distinctive specific cell answers. Although no SARM drug candidate (aiming for tes...

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Identifiers and source

Literature Corpus work
1896a495-7c01-50c4-9d81-9d15864d0f4e
DOI
10.1016/j.jevs.2012.01.005
Open publication

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Characterization of In Vitro Synthesized Equine Metabolites of the Selective Androgen Receptor Modulators S24 and S4DOI 10.1016/j.jevs.2012.01.005
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