Article

Target class profiling of small molecule methyltransferases

2022-03-24

Abstract excerpt

Target class profiling (TCP) is a chemical biology approach to investigating understudied biological target classes. TCP is achieved by developing a generalizable assay platform and screening curated compound libraries to interrogate the chemical biological space of members of an enzyme family with clinical and biological importance. In this work we took a TCP approach to investigate inhibitory activity across a s...

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Identifiers and source

Literature Corpus work: e9086394-c485-5d81-8d7b-b0c78bc3070d
DOI: 10.1101/2022.03.24.485659

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