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Article

Differential desensitization of dopamine D2 receptor isoforms by protein kinase C: the importance of receptor phosphorylation and pseudosubstrate sites.

European journal of pharmacology - 22 Dec 2007

Morris Stephen J, Van-Ham Irit Itzhaki, Daigle Mireille, Robillard Liliane, Sajedi Naghmeh, Albert Paul R

Abstract excerpt

Altered regulation of dopamine D(2) receptors is implicated in addiction, schizophrenia and movement disorders, as well as lactotroph growth and regulation. Dopamine D(2S) and dopamine D(2L) receptors are alternately-spliced variants that differ by 29 amino acids in the third intracellular (i3) d...

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Identifiers

PMID: 17869243
DOI: 10.1016/j.ejphar.2007.08.027

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PubMed metadata and Literature Corpus relationships. Corpus snapshot updated 2 Sept 2026. Prepared record publication-17869243-2026-09-02.2. Manifest publication-graph-cohort-2026-09-02.2.

Source receipt: PubMed via Helena Literature Corpus, retrieved 2 Sept 2026.

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