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Arylazolyl(azinyl)thioacetanilide. Part 9: Synthesis and biological investigation of thiazolylthioacetamides derivatives as a novel class of potential antiviral agents.

Archives of pharmacal research - 1 Jun 2012

Zhan Peng, Wang Liu, Liu Hong, Chen Xuwang, Li Xiao, Jiang Xin, Zhang Qiangqiang, Liu Xinyong, Pannecouque Christophe, Naesens Lieve, De Clercq Erik, Liu Ailin, Du Guanhua

Abstract excerpt

In continuation of our endeavor to develop new, potent, selective and less toxic antiviral agents, a novel series of 2-(2-amino/chloro-4-(2,4-dibromophenyl) thiazol-5-ylthio)acetamide derivatives was synthesized via an expeditious route and evaluated for their anti-HIV activities against wild-type virus and clinically relevant mutant strains, and for their anti-influenza virus activities against influenza A (H1N1...

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PMID: 22870806
DOI: 10.1007/s12272-012-0604-y

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PubMed metadata and Literature Corpus relationships. Corpus snapshot updated 7 Sept 2026. Manifest publication-graph-cohort-2026-09-07.1.

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