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Article

Agonist binding to peptide hormone receptors.

Biochemical Society transactions - 1 Feb 2003

Wheatley M, Hawtin S R, Wesley V J, Howard H C, Simms J, Miles A, McEwan K, Parslow R A

Abstract excerpt

A fundamental issue in molecular pharmacology is to define how agonist-receptor interaction differs from that of antagonist-receptor interaction. The V(1a) vasopressin receptor (V(1a)R) is a member of a family of related G-protein-coupled receptors (GPCRs) that are activated by vasopressin, oxytocin (OT) and related peptides. A segment of the N-terminus that was required for agonist binding, but not antagonist...

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Identifiers

PMID: 12546649
DOI: 10.1042/bst0310035

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PubMed metadata and Literature Corpus relationships. Corpus snapshot updated 7 Sept 2026. Manifest publication-graph-cohort-2026-09-08.1.

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