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Article

Real-time analysis of dopamine: antagonist interactions at recombinant human D2long receptor upon modulation of its activation state.

British journal of pharmacology - 1 Sept 2001

Pauwels P J, Tardif S, Wurch T, Colpaert F C

Abstract excerpt

1. Antipsychotic drugs may mediate their therapeutic effects not only by preventing the binding of dopamine but also by decreasing the propensity of the dopamine receptor to assume an active R* state. Ligand-mediated activation and blockade of the recombinant human D(2long) receptor was investiga...

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Identifiers

PMID: 11522600
DOI: 10.1038/sj.bjp.0704243
PMCID: PMC1572932

Provenance

PubMed metadata and Literature Corpus relationships. Corpus snapshot updated 1 Sept 2026. Prepared record publication-11522600-2026-09-01.1. Manifest publication-graph-cohort-2026-09-01.1.

Source receipt: PubMed via Helena Literature Corpus, retrieved 1 Sept 2026.

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