Article
Insights into matriptase-2 substrate binding and inhibition mechanisms by analyzing active-site-mutated variants.
ChemMedChem - 2 Jan 2012
Maurer Eva, Sisay Mihiret T, Stirnberg Marit, Steinmetzer Torsten, Bajorath Jürgen, Gütschow Michael
Abstract excerpt
No abstract is available from the source.
Topics
- Amino Acid Sequence
- Catalytic Domain
- HEK293 Cells
- Humans
- Membrane Proteins
- Models, Molecular
- Mutagenesis, Site-Directed
- Mutation
- Peptides
- Protease Inhibitors
- Serine Endopeptidases
- Substrate Specificity
