Discover Community Create You

Loading publication...

Noodle always counts identifier-free feature events for service operation. With your permission, Google Analytics can also estimate audience and engagement. Search text, publication identifiers, cookies, IP addresses and browser fingerprints are never included in Noodle's first-party event counters.

Privacy details

Article

Design and synthesis of cyclic sulfonamides and sulfamates as new calcium sensing receptor agonists.

Bioorganic & medicinal chemistry letters - 15 Dec 2010

Kiefer Lionel, Gorojankina Tatiana, Dauban Philippe, Faure Hélène, Ruat Martial, Dodd Robert H

Abstract excerpt

The design, synthesis and calcimimetic properties of various cyclic sulfonamides and sulfamates are described. The latter were prepared from the corresponding o-alkenylarenesulfonamides via copper- or rhodium-catalyzed intramolecular aziridination. The size of the cyclic sulfonamide rings as well...

Read the complete abstract on PubMed

Topics

Share this publication in a Topic to start or enrich a Post.

Share to Copper
Share to Cyclization
Share to Drug Design

Methodology Data sources Editorial policy Privacy About Contact Helena Bioinformatics

Share to Molecular Conformation

Share to Receptors, Calcium-Sensing

Share to Stereoisomerism

Share to Sulfonamides

Share to Sulfonic Acids

Source

Identifiers

PMID: 21041081
DOI: 10.1016/j.bmcl.2010.10.006

Provenance

PubMed metadata and Literature Corpus relationships. Corpus snapshot updated 2 Sept 2026. Prepared record publication-21041081-2026-09-02.2. Manifest publication-graph-cohort-2026-09-02.2.

Source receipt: PubMed via Helena Literature Corpus, retrieved 2 Sept 2026.

Related research

Semantic proximity does not establish scientific evidence.

Research trail→

Click a neighbor to travelStep 1 · 8 closest

Design and synthesis of cyclic sulfonamides and sulfamates as new calcium sensing receptor agonists.PMID 21041081Read ↗

Next-Generation Analogues of AC265347 as Positive Allosteric Modulators of the Calcium-Sensing Receptor: Pharmacological Investigation of Structural Modifications at the Stereogenic CentreSemantic proximity Read ↗

Structure-activity studies on arylamides and arysulfonamides Ras inhibitors.Semantic proximity Read ↗

Anthranilic sulfonamide CCK1/CCK2 dual receptor antagonists I: discovery of CCKR1 selectivity in a previously CCKR2-selective lead series.Semantic proximity Read ↗

(2E)-5-[3-[(phenylsulfonyl)amino]phenyl]-pent-2-en-4-ynohydroxamic acid and its derivatives as novel and potent inhibitors of ras transformation.Semantic proximity Read ↗

Transient Sulfenic Acids in the Synthesis of Biologically Relevant ProductsSemantic proximity Read ↗

Solution-phase parallel synthesis of carbamates as gamma-secretase inhibitors.Semantic proximity Read ↗

Syntheses and biological properties of cysteine-reactive epibatidine derivatives.Semantic proximity Read ↗

Synthesis and biological activity of new iodoacetamide derivatives on mutants of squalene-hopene cyclase.Semantic proximity Read ↗

⌁Select a neighboring publication to make it the new centre.