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Article

A series of C-terminal amino alcohol dipeptide A beta inhibitors.

Bioorganic & medicinal chemistry letters - 4 Nov 2002

Garofalo Albert W, Wone David W G, Phuc Angela, Audia James E, Bales Cheryl A, Dovey Harry F, Dressen Darren B, Folmer Beverly, Goldbach Erich G, Guinn Ashley C, Latimer Lee H, Mabry Thomas E, Nissen Jeffrey S, Pleiss Michael A, Sohn Stephen, Thorsett Eugene D, Tung Jay S, Wu Jing

Abstract excerpt

Potent, small molecule A beta inhibitors have been prepared that incorporate an alanine core bracketed by an N-terminal arylacetyl group and various C-terminal amino alcohols. The compounds exhibit stereospecific inhibition as demonstrated in an in vitro assay.

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Methodology Data sources Editorial policy Privacy About Contact Helena Bioinformatics

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Identifiers

PMID: 12372499
DOI: 10.1016/s0960-894x(02)00684-4

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PubMed metadata and Literature Corpus relationships. Corpus snapshot updated 7 Sept 2026. Manifest publication-graph-cohort-2026-09-07.1.

Source receipt: pubmed, retrieved 7 Sept 2026.

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