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Article

A multidisciplinary approach for the identification of novel HIV-1 non-nucleoside reverse transcriptase inhibitors: S-DABOCs and DAVPs.

ChemMedChem - 1 Apr 2008

Radi Marco, Falciani Chiara, Contemori Lorenzo, Petricci Elena, Maga Giovanni, Samuele Alberta, Zanoli Samantha, Terrazas Montserrat, Castria Marinunzia, Togninelli Andrea, Esté José A, Clotet-Codina Imma, Armand-Ugón Mercedes, Botta Maurizio

Abstract excerpt

Among the FDA approved drugs for the treatment of AIDS, non-nucleoside reverse transcriptase inhibitors (NNRTIs) are essential components of first-line anti-HIV-1 therapy because of the less-severe adverse effects associated with NNRTIs administration in comparison to therapies based on other anti-HIV-1 agents. In this contest, 3,4-dihydro-2-alkoxy-6-benzyl-4-oxypyrimidines (DABOs) have been the object of many...

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Identifiers

PMID: 18081133
DOI: 10.1002/cmdc.200700198

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PubMed metadata and Literature Corpus relationships. Corpus snapshot updated 7 Sept 2026. Manifest publication-graph-cohort-2026-09-07.1.

Source receipt: pubmed, retrieved 7 Sept 2026.

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